Regulatory Protein Expression Vectors

We offer several regulatory protein or partner protein expression vectors that are used in NanoBRET® Intracellular Kinase Target Engagement (TE) Assays.

For kinases requiring co-expression of a regulatory or partner protein, the expression vector is co-transfected with the appropriate kinase-NanoLuc® fusion vector prior to performing the NanoBRET® Kinase TE Assay. The "Used in Kinase TE Assay" column in the table below provides links to application notes with example data and assay details.

Search by Regulator Name
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Regulator Regulator Plasmid Name Cat.# Used in Kinase TE Assay
CCNA1 CCNA1 Expression Vector NV2591 CDK2/Cyclin A1
CCNB1 CCNB1 Expression Vector NV2601 CDK1/Cyclin B1
CCNC CCNC Expression Vector NV2611 CDK8/Cyclin C; CDK19/Cyclin C
CCND1 CCND1 Expression Vector NV2621 CDK4/Cyclin D1; CDK6/Cyclin D1
CCND3 CCND3 Expression Vector NV2631 CDK4/Cyclin D3
CCNE1 CCNE1 Expression Vector NV2641 CDK1/Cyclin E1; CDK2/Cyclin E1; CDK3/Cyclin E1
CCNH CCNH Expression Vector NV2651 CDK20/Cyclin H
CCNK CCNK Expression Vector NV2661 CDK9/Cyclin K/K-8; CDK9/Cyclin K/K-10; CDK11A/Cyclin K; CDK11B/Cyclin K
CCNL2 CCNL2 Expression Vector NV2671 CDK10/Cyclin L2; CDK11A/Cyclin L2; CDK11B/Cyclin L2
CCNT1 CCNT1 Expression Vector NV2681 CDK9/Cyclin T1
CCNY CCNY Expression Vector NV2691 CDK14/Cyclin Y; CDK15/Cyclin Y; CDK16/Cyclin Y; CDK17/Cyclin Y; CDK18/Cyclin Y
CDK5R1 CDK5R1 Expression Vector NV2821 CDK5/CDK5R1
CDK5R2 CDK5R2 Expression Vector NV2831 CDK5/CDK5R2
PIK3R1 PIK3R1 Expression Vector NV4031 PIK3CA/PIK3R1; PIK3CA(C420R)/PIK3R1; PIK3CA(E542K)/PIK3R1; PIK3CA(E545A)/PIK3R1; PIK3CA(E545K)/PIK3R1; PIK3CA(Q546K)/PIK3R1; PIK3CA(I800L)/PIK3R1; PIK3CA(M1043I)/PIK3R1; PIK3CA(H1047L)/PIK3R1; PIK3CA(H1047R)/PIK3R1; PIK3CA(H1047Y)/PIK3R1, PIK3CB/PIK3R1; PIK3CD/PIK3R1

Assays available for over 340+ kinases

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